Affinity DataKi: 0.0700nMAssay Description:Inhibitory activity against human tryptase enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibitory activity against human tryptase enzymeMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Inhibitory activity against human mast cell tryptase betaMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibitory activity against human mast cell tryptase betaMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
Affinity DataKi: 3.25nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 3.75nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 4nMAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
Affinity DataKi: 4.30nMAssay Description:Inhibitory activity against human mast cell tryptase betaMore data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 5nM ΔG°: -11.2kcal/molepH: 8.2 T: 2°CAssay Description:Enzymes were incubated with inhibitors at eight inhibitor concentrations bracketing the Ki, prepared by serial dilution along with control lacking th...More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Binding affinity to human tryptase beta2More data for this Ligand-Target Pair
Affinity DataKi: 5.40nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 5.80nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
Affinity DataKi: 6.20nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:In vitro inhibition of human Tryptase beta.More data for this Ligand-Target Pair
Affinity DataKi: 6.55nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 7.60nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 9.20nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 9.60nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 9.80nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibitory activity against human Tryptase beta was evaluatedMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Inhibitory potency against tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Inhibitory activity against human Tryptase beta was evaluatedMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:In vitro inhibition of human Tryptase beta.More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:In vitro inhibition of human Tryptase beta.More data for this Ligand-Target Pair
Affinity DataKi: 21nMAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:In vitro inhibition of human Tryptase beta.More data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Inhibition of human B tryptaseMore data for this Ligand-Target Pair
Affinity DataKi: 23nM ΔG°: -10.3kcal/molepH: 7.4 T: 2°CAssay Description:Each enzyme was assayed with a set of different concentrations of each inhibitor. After addition of the appropriate substrate, the rate of hydrolysis...More data for this Ligand-Target Pair